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Paper Title
Discovery of LSZ102, a Potent, Orally Bioavailable Selective Estrogen Receptor Degrader (SERD) for the Treatment of Estrogen Receptor Positive Breast Cancer.
PubMed
Paper Journal Title
J Med Chem
Paper Citation Count
71
Paper Publication Year
2018
Bio Mention
ER, ER positive breast cancer, Estrogen, Estrogen Receptor, Estrogen Receptor Positive Breast Cancer, LSZ102, SERDs, aromatase, benzothiophene, breast cancer, estrogen, estrogen receptor, estrogen receptor alpha, estrogen receptor alpha (, fulvestrant, patients, steroid
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Author Name
Affiliation
Sunkyu Kim
Novartis Institutes for BioMedical Research, Inc.
Donald P McDonnell
Duke University School of Medicine
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