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Paper Details

Discovery of Competitive and Noncompetitive Ligands of the Organic Cation Transporter 1 (OCT1; SLC22A1).
J Med Chem
43
2017
1-benzyl-1,2,3,4-tetrahydroisoquinoline, ASP, OCT1, Organic Cation Transporter 1, Organic cation transporter 1, SLC22A1, eukaryotic homologue, human, human OCT1
Drug Discovery, HEK293 Cells, Humans, Ligands, Molecular Docking Simulation, Organic Cation Transporter 1, Small Molecule Libraries
Author NameAffiliation
Eugene C ChenUniversity of California san francisco
Natalia KhuriUniversity of California san francisco
Xiaomin LiangUniversity of California san francisco
Adrian SteculaUniversity of California san francisco
Huan-Chieh ChienUniversity of California san francisco
Sook Wah YeeUniversity of California san francisco
Yong Huang
Andrej Sali (CM4AI)University of California san francisco
Andrej Sali (CM4AI)California Institute of Quantitative Biosciences, University of California san francisco
Andrej Sali (CM4AI)Department of Pharmaceutical Chemistry, University of California san francisco
Andrej Sali (CM4AI)University of California san francisco
Andrej Sali (CM4AI)Department of Pharmaceutical Chemistry, University of California san francisco
Andrej Sali (CM4AI)California Institute of Quantitative Biosciences, University of California san francisco
Kathleen M GiacominiUniversity of California san francisco
Kathleen M GiacominiDepartment of Pharmaceutical Chemistry, University of California san francisco
Kathleen M GiacominiCalifornia Institute of Quantitative Biosciences, University of California san francisco
Kathleen M GiacominiInstitute of Human Genetics, University of California san francisco
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