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Paper Details

Fragment binding to the Nsp3 macrodomain of SARS-CoV-2 identified through crystallographic screening and computational docking.
Sci Adv
96
2021
Nsp3 macrodomain, SARS, SARS-CoV, SARS-CoV-2, SARS-CoV-2 macrodomain, active site, adenosine diphosphate, macrodomain, nonstructural protein 3, severe, severe acute respiratory syndrome
Author NameAffiliation
Galen J CorreyUniversity of California San Francisco
Iris D YoungUniversity of California San Francisco
Iris D YoungQuantitative Biosciences Institute (QBI) Coronavirus Research Group Structural Biology Consortium, University of California San Francisco
Ursula Schulze-GahmenQuantitative Biosciences Institute (QBI) Coronavirus Research Group Structural Biology Consortium, University of California San Francisco
Tristan W OwensQuantitative Biosciences Institute (QBI) Coronavirus Research Group Structural Biology Consortium, University of California San Francisco
Ishan DeshpandeQuantitative Biosciences Institute (QBI) Coronavirus Research Group Structural Biology Consortium, University of California San Francisco
Gregory E MerzQuantitative Biosciences Institute (QBI) Coronavirus Research Group Structural Biology Consortium, University of California San Francisco
Justin T BielQuantitative Biosciences Institute (QBI) Coronavirus Research Group Structural Biology Consortium, University of California San Francisco
Jessica K PetersQuantitative Biosciences Institute (QBI) Coronavirus Research Group Structural Biology Consortium, University of California San Francisco
Michelle MoritzQuantitative Biosciences Institute (QBI) Coronavirus Research Group Structural Biology Consortium, University of California San Francisco
Nadia HerreraQuantitative Biosciences Institute (QBI) Coronavirus Research Group Structural Biology Consortium, University of California San Francisco
Huong T KratochvilQuantitative Biosciences Institute (QBI) Coronavirus Research Group Structural Biology Consortium, University of California San Francisco
James M Holton
James M HoltonUniversity of California San Francisco
James M HoltonLawrence Berkeley National Laboratory
Natalia JuraUniversity of California San Francisco
Alan AshworthUniversity of California San Francisco
John J IrwinDepartment of Pharmaceutical Chemistry, University of California San Francisco
Michael C ThompsonUniversity of California Merced
Jason E GestwickiDepartment of Pharmaceutical Chemistry, University of California San Francisco
Jason E GestwickiInstitute for Neurodegenerative Disease, University of California San Francisco
Brian K ShoichetDepartment of Pharmaceutical Chemistry, University of California San Francisco
Brian K ShoichetDepartment of Pharmaceutical Chemistry, University of California San Francisco
James S FraserUniversity of California San Francisco
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