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Paper Title
Structure-based ligand discovery for the Large-neutral Amino Acid Transporter 1, LAT-1.
PubMed
Paper Journal Title
Proc Natl Acad Sci U S A
Paper Citation Count
135
Paper Publication Year
2013
Bio Mention
Amino Acid, LAT-1, Large-neutral Amino Acid Transporter 1, acivicin, amino acids, cancer, cancer cell line, drug, sodium
Mesh Descriptor
Amines, Analysis of Variance, Blood-Brain Barrier, Cell Line, Tumor, Crystallography, X-Ray, Cyclohexanecarboxylic Acids, Drug Delivery Systems, Flow Cytometry, Gabapentin, Glioblastoma, HEK293 Cells, Humans, Isoxazoles, Large Neutral Amino Acid-Transporter 1, Leucine, Ligands, Models, Molecular, Tritium, gamma-Aminobutyric Acid
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Ethan G Geier
University of California san francisco
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