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Paper Details

Small-Molecule Allosteric Modulators of the Protein Kinase PDK1 from Structure-Based Docking.
J Med Chem
18
2015
PDK1, PIF, PIF pocket, Protein Kinase PDK1, allosteric, allosteric peptide
3-Phosphoinositide-Dependent Protein Kinases, Allosteric Site, Computer Simulation, Crystallography, X-Ray, Dose-Response Relationship, Drug, High-Throughput Screening Assays, Humans, Models, Molecular, Molecular Docking Simulation, Protein Binding, Small Molecule Libraries, Structure-Activity Relationship
Author NameAffiliation
Terry J RettenmaierUniversity of California san francisco
Terry J RettenmaierDepartment of Pharmaceutical Chemistry, University of California san francisco
Hao FanDepartment of Pharmaceutical Chemistry, University of California san francisco
Hao FanBioinformatics Institute (BII)
Hao FanNational University of Singapore
Joel KarpiakUniversity of California san francisco
Joel KarpiakDepartment of Pharmaceutical Chemistry, University of California san francisco
Allison K DoakDepartment of Pharmaceutical Chemistry, University of California san francisco
Andrej Sali (CM4AI)University of California san francisco
Andrej Sali (CM4AI)University of California san francisco
Brian K ShoichetDepartment of Pharmaceutical Chemistry, University of California san francisco
Brian K ShoichetDepartment of Pharmaceutical Chemistry, University of California san francisco
James A WellsDepartment of Pharmaceutical Chemistry, University of California san francisco
James A WellsUniversity of California san francisco
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