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Paper Title
Translation Termination Factor GSPT1 Is a Phenotypically Relevant Off-Target of Heterobifunctional Phthalimide Degraders.
PubMed
Paper Journal Title
ACS Chemical Biology
Paper Citation Count
99
Paper Publication Year
2018
Bio Mention
CRBN, CRL4CRBN, CUL4, DDB1, E3 ligase, G1 to S phase transition 1, GSPT1, PHA665752, Phthalimide, RBX1, RTKs, Translation Termination Factor GSPT1, leukemia, leukemia cell lines, phthalimide, receptor tyrosine kinases, sunitinib, targeting, translation termination factor, tyrosine
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Author Name
Affiliation
James E Bradner
Dana-Farber Cancer Institute
James E Bradner
Novartis Institutes for Biomedical Research
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