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Sulfopin is a covalent inhibitor of Pin1 that blocks Myc-driven tumors in vivo.
Nat Chem Biol
64
2021
Cys113, MYCN, MYCN-driven neuroblastoma, Myc, Pin1, Sulfopin, active, c-Myc target genes, cancer, cancer cell line, cells, murine, oncogenes, pancreatic cancer, peptidyl-prolyl isomerase, prolyl, tumor, tumor suppressors, tumors, zebrafish
Author NameAffiliation
Sirano Dhe-PaganonDana-Farber Cancer Institute
Alex LookDana-Farber Cancer Institute, Harvard Medical School
Alex LookDivision of Pediatric Hematology/Oncology Boston Children's Hospital
Rosalie C SearsOregon Health & Science University
Rosalie C SearsBrenden-Colson Center for Pancreatic Care, Oregon Health & Science University
Rosalie C SearsKnight Cancer Institute, Oregon Health & Science University
Rosalie C SearsOregon Health & Science University
Rosalie C SearsKnight Cancer Institute, Oregon Health & Science University
Rosalie C SearsBrenden-Colson Center for Pancreatic Care, Oregon Health & Science University
Nathanael S GrayDana-Farber Cancer Institute
Nathanael S GrayChem-H and Stanford Cancer Institute, Stanford School of Medicine, Stanford University
Nathanael S GrayHarvard Medical School
Nathanael S GrayDana-Farber Cancer Institute
Nathanael S GrayHarvard Medical School
Nathanael S GrayChem-H and Stanford Cancer Institute, Stanford School of Medicine, Stanford University
Nir LondonThe Weizmann Institute of Science
Nir LondonThe Weizmann Institute of Science
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