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Paper Title
Computational Discovery and Experimental Validation of Inhibitors of the Human Intestinal Transporter OATP2B1.
PubMed
Paper Journal Title
J Chem Inf Model
Paper Citation Count
13
Paper Publication Year
2017
Bio Mention
Human, Human Intestinal Transporter OATP2B1, OATP member 2B1 transporter, OATP2B1, OATP2B1 transporter, OATPs, bicalutamide, estrone-3-sulfate, intestinal OATP2B1, meloxicam, organic anion transporters, ticagrelor
Mesh Descriptor
Animals, CHO Cells, Computer Simulation, Cricetinae, Cricetulus, Drug Discovery, Drug Evaluation, Preclinical, Humans, Inhibitory Concentration 50, Molecular Docking Simulation, Organic Anion Transporters, Protein Conformation
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Author Name
Affiliation
Natalia Khuri
Stanford University
Andrej Sali (CM4AI)
Department of Pharmaceutical Chemistry and California Institute of Quantitative Biosciences (QB3), University of California San Francisco
Andrej Sali (CM4AI)
Department of Pharmaceutical Chemistry and California Institute of Quantitative Biosciences (QB3), University of California San Francisco
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