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Paper Details

Functional TRIM24 degrader via conjugation of ineffectual bromodomain and VHL ligands.
Nat Chem Biol
148
2018
TRIM24, TRIM24 bromodomain, VHL, VHL E3 ubiquitin ligase, VHL ligands, acute leukemia, bromodomain, cancer, cancers, chromatin, dTRIM24
Author NameAffiliation
Mousheng XuDana-Farber Cancer Institute
Sirano Dhe-PaganonDana-Farber Cancer Institute
Jun QiDana-Farber Cancer Institute
Jun QiHarvard Medical School
Nathanael S GrayDana-Farber Cancer Institute
Nathanael S GrayHarvard Medical School
Nathanael S GrayDana-Farber Cancer Institute
Nathanael S GrayHarvard Medical School
James E BradnerDana-Farber Cancer Institute
James E BradnerHarvard Medical School
James E BradnerNovartis Institutes for Biomedical Research
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