|
| 37169961 | Signal peptide mimicry primes Sec61 for client-selective inhibition. | Nat Chem Biol | 2023 |
| 35434798 | Inhibition of the Sec61 translocon overcomes cytokine-induced glucocorticoid resistance in T-cell acute lymphoblastic leukaemia. | Br J Haematol | 2022 |
| 33592144 | Inhibitors of Eukaryotic Translational Machinery as Therapeutic Agents. | J Med Chem | 2021 |
| 32353859 | A SARS-CoV-2 protein interaction map reveals targets for drug repurposing. | Nature | 2020 |
| 31742404 | Total Syntheses of the 3<i>H</i>-Pyrrolo[2,3-<i>c</i>]quinolone-Containing Alkaloids Marinoquinolines A-F, K, and Aplidiopsamine A Using a Palladium-Catalyzed Ullmann Cross-Coupling/Reductive Cyclization Pathway. | J Org Chem | 2020 |
| 30281974 | Mechanistic Studies on the Base-Promoted Conversion of Alkoxy-Substituted, Ring-Fused gem-Dihalocyclopropanes into Furans: Evidence for a Process Involving Electrocyclic Ring Closure of a Carbonyl Ylide Intermediate. | J Org Chem | 2018 |
| 29259751 | Design, Synthesis, and Biological Activity of 1,2,3-Triazolobenzodiazepine BET Bromodomain Inhibitors. | ACS Med Chem Lett | 2017 |
| 28451332 | Synthesis of rhamnosylated arginine glycopeptides and determination of the glycosidic linkage in bacterial elongation factor P. | Chem Sci | 2017 |
| 28320614 | Synthesis of a GlcNAcylated arginine building block for the solid phase synthesis of death domain glycopeptide fragments. | Bioorg Med Chem | 2017 |
| 27055867 | BET inhibition represses miR17-92 to drive BIM-initiated apoptosis of normal and transformed hematopoietic cells. | Leukemia | 2016 |
| 27213690 | CIS is a potent checkpoint in NK cell-mediated tumor immunity. | Nat Immunol | 2016 |
| 25778803 | A RIPK2 inhibitor delays NOD signalling events yet prevents inflammatory cytokine production. | Nat Commun | 2015 |
| 25944566 | BET inhibitors induce apoptosis through a MYC independent mechanism and synergise with CDK inhibitors to kill osteosarcoma cells. | Sci Rep | 2015 |
| 24261714 | BET bromodomain inhibitors: a patent review. | Expert Opin Ther Pat | 2014 |
| 24677741 | Simplified silvestrol analogues with potent cytotoxic activity. | ChemMedChem | 2014 |
| 23692341 | Consecutive gold(I)-catalyzed cyclization reactions of o-(buta-1,3-diyn-1-yl-)-substituted N-aryl ureas: a one-pot synthesis of pyrimido[1,6-a]indol-1(2H)-ones and related systems. | Org Lett | 2013 |