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| 35753676 | Chemical biology and pharmacology of histone lysine methylation inhibitors. | Biochim Biophys Acta Gene Regul Mech | 2022 |
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| 35907431 | Enzymatic nucleosome acetylation selectively affects activity of histone methyltransferases in vitro. | Biochim Biophys Acta Gene Regul Mech | 2022 |
| 36084291 | Combinatorial Anticancer Drug Screen Identifies Off-Target Effects of Epigenetic Chemical Probes. | ACS Chem Biol | 2022 |
| 34164919 | Development of LM98, a Small-Molecule TEAD Inhibitor Derived from Flufenamic Acid. | ChemMedChem | 2021 |
| 33522809 | Discovery of Small-Molecule Antagonists of the PWWP Domain of NSD2. | J Med Chem | 2021 |
| 33742187 | Protein arginine methylation: from enigmatic functions to therapeutic targeting. | Nat Rev Drug Discov | 2021 |
| 33513288 | Rational Design and Synthesis of Selective PRMT4 Inhibitors: A New Chemotype for Development of Cancer Therapeutics*. | ChemMedChem | 2021 |
| 33591753 | A First-in-Class, Highly Selective and Cell-Active Allosteric Inhibitor of Protein Arginine Methyltransferase 6. | J Med Chem | 2021 |
| 33579912 | PRMT5 inhibition disrupts splicing and stemness in glioblastoma. | Nat Commun | 2021 |
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| 34154424 | Discovery of the SMYD3 Inhibitor BAY-6035 Using Thermal Shift Assay (TSA)-Based High-Throughput Screening. | SLAS Discov | 2021 |
| 33980013 | Design, Synthesis, and Evaluation of WD-Repeat-Containing Protein 5 (WDR5) Degraders. | J Med Chem | 2021 |
| 32367723 | Discovery of a First-in-Class Protein Arginine Methyltransferase 6 (PRMT6) Covalent Inhibitor. | J Med Chem | 2020 |
| 33054974 | Correction: A chemical probe of CARM1 alters epigenetic plasticity against breast cancer cell invasion. | Elife | 2020 |
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| 32297856 | Telomere dysfunction cooperates with epigenetic alterations to impair murine embryonic stem cell fate commitment. | Elife | 2020 |
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| 30352278 | Characterization of inv(3) cell line OCI-AML-20 with stroma-dependent CD34 expression. | Exp Hematol | 2019 |
| 31781029 | Synthetic Peptides as Therapeutic Agents: Lessons Learned From Evolutionary Ancient Peptides and Their Transit Across Blood-Brain Barriers. | Front Endocrinol (Lausanne) | 2019 |
| 31657716 | A chemical probe of CARM1 alters epigenetic plasticity against breast cancer cell invasion. | Elife | 2019 |
| 31848333 | Discovery of a chemical probe for PRDM9. | Nat Commun | 2019 |
| 31559307 | SETD7 at the heart of chromatin factor interplay. | Stem Cell Investig | 2019 |
| 31415173 | Selective, Small-Molecule Co-Factor Binding Site Inhibition of a Su(var)3-9, Enhancer of Zeste, Trithorax Domain Containing Lysine Methyltransferase. | J Med Chem | 2019 |
| 31408619 | Therapeutic Targeting of RNA Splicing Catalysis through Inhibition of Protein Arginine Methylation. | Cancer Cell | 2019 |
| 31287992 | A C19MC-LIN28A-MYCN Oncogenic Circuit Driven by Hijacked Super-enhancers Is a Distinct Therapeutic Vulnerability in ETMRs: A Lethal Brain Tumor. | Cancer Cell | 2019 |
| 31260300 | Discovery of a Potent and Selective Fragment-like Inhibitor of Methyllysine Reader Protein Spindlin 1 (SPIN1). | J Med Chem | 2019 |
| 31285596 | Fragment-based discovery of a chemical probe for the PWWP1 domain of NSD3. | Nat Chem Biol | 2019 |
| 30926792 | Targeting bivalency de-represses Indian Hedgehog and inhibits self-renewal of colorectal cancer-initiating cells. | Nat Commun | 2019 |
| 30774623 | Teneurin C-Terminal Associated Peptide (TCAP)-1 and Latrophilin Interaction in HEK293 Cells: Evidence for Modulation of Intercellular Adhesion. | Front Endocrinol (Lausanne) | 2019 |
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| 30462309 | Direct interaction between the PRDM3 and PRDM16 tumor suppressors and the NuRD chromatin remodeling complex. | Nucleic Acids Res | 2019 |
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